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| 产地 | 中国 |
| 品牌 | 爱必信(absin) |
| 货号 | abs816033 |
| 用途 | 见爱必信官网 |
| 包装规格 | 50mg,50mg,200mg,200mg,500mg,500mg |
| 纯度 | 99%% |
| CAS编号 | 152-11-4 |
| 别名 | 盐酸维拉帕米;(±)-Verapamil hydrochlorid |
| 是否进口 | 否 |
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抑制剂描述: 产品名称:Verapamil hydrochloride 产品别名:见爱必信官网 英文别名:Verapamil hydrochloride 靶点:Calcium Channel CAS:152-11-4 纯度:99% 外观:见爱必信官网 保存方法:Store at -20℃ for one year(Powder);Store at 2-4℃ for two weeks;Store at -20℃ for six months after dissolution. 描述: 溶解性:DMSO :98mg/mL(199.56mM) 体外研究:
The enzyme hydrolase activity of recombinant CES2 is substantially inhibited by diltiazem and verapamil (Ki = 0.25 ± 0.02 and 3.84 ± 0.99μM, respectively). 体内研究:Verapamil confers an anti-arrhythmic effect via calcium influx inhibition, inhibition of oxygen consumption and accompanied by preservation of Cx43 protein in rat heart.
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