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试剂描述:

产品名称:MEK Inhibitor I

产品别名:

CAS号:297744-42-4

英文别名:MEK Inhibitor I

分子量:374.46

分子式:C₂₁H₁₈N₄OS

纯度:≥95%

外观:见爱必信官网

保存方法:Store at -20° C

描述:MEK Inhibitor I is a cell-permeable, pyridine-containing, vinylogous cyanamide that has the ability to act as a selective and potent inhibitor of MEK with little activity towards MKK3 and MKK4. The compound displays significant affinity only towards ATP-bound MEK (i.e. noncompetitive with respect to ATP) and the demonstrated inhibition is noncompetitive with respect to ERK. Compared to U0126 in aqueous solutionsMEK Inhibitor I demonstrates superior potency, solubility, and stability. Additionally shown to protect against phorbol ester-mediated ear edema in mice.

应用:A vinylogous cyanamide that has the ability to act as a selective and potent inhibitor of MEK

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